Compound name
SGC-GAK-1N
Protein family
Protein Kinase
Target name
GAK
Affinity on-target cellular (nM)
5000
CG-Set
Kinase set
Recommended Concentration
1 µM
Compound EUbOPEN ID
EUB0000229b
SMILES
COc1cc(N(C)c2ccnc3ccc(C(F)(F)F)cc23)cc(OC)c1OC
InChIKey
PVTQCCFMFWASHK-UHFFFAOYSA-N
NCBI gene ID
2580
UniProt ID
O14976
Synonyms
DNAJC26
Mode of action
Negative control for SGC-GAK-1
Affinity on-target cellular definition
IC50
Affinity on-target cellular assay type
NanoBRET assay (HEK293T cells)
Affinity on-target cellular source knowledge
https://pubs.acs.org/doi/10.1021/acs.jmedchem.8b01213
Affinity on-target cellular relation
>