Compound name
PPTN
Protein family
GPCR
Target name
P2RY14
Affinity biochemical (nM)
7.94
Compound EUbOPEN ID
EUB0000274cCl
SMILES
Cl.OC(=O)c1cc(-c2ccc(cc2)C2CCNCC2)c2ccc(cc2c1)-c1ccc(cc1)C(F)(F)F
InChIKey
FKMVYPCBLWYNAV-UHFFFAOYSA-N
NCBI gene ID
9934
UniProt ID
Q15391
Synonyms
KIAA0001
Mode of action
Antagonist
Affinity biochemical definition
IC50
Affinity biochemical assay type
Antagonist activity human P2Y14R expressed in African green monkey COS7 cells assessed as inhibition of UDPG-induced [3H]inositol phosphate accumulation after 30 mins by liquid scintillation counting method
Affinity Biochemical Source Knowledge
27331270
Affinity biochemical relation
=