Compound name
BRL-52537
Protein family
GPCR
Target name
OPRK1
Affinity on-target cellular (nM)
10.96
Compound EUbOPEN ID
EUB0000365aCl
SMILES
[H]Cl.O=C(CC1=CC(Cl)=C(Cl)C=C1)N2CCCC[C@H]2CN3CCCC3
InChIKey
NGVLSOWJSUUYDE-RSAXXLAASA-N
NCBI gene ID
4986
UniProt ID
P41145
Synonyms
KOR, OPRK
Mode of action
Agonist
Affinity on-target cellular definition
IC50
Affinity on-target cellular assay type
Kappa-opioid receptor agonist potency in vitro using rabbit vas deferens(LVD) preparation
Affinity on-target cellular relation
=