Compound name
DEXMEDETOMIDINE
Protein family
GPCR
Target name
ADRA2A
Affinity on-target cellular (nM)
1.51
Compound EUbOPEN ID
EUB0000404aCl
SMILES
[H]Cl.C[C@H](C1=CN=CN1)C1=C(C)C(C)=CC=C1
InChIKey
VPNGEIHDPSLNMU-MERQFXBCSA-N
NCBI gene ID
150
UniProt ID
P08913
Synonyms
ADRAR
Affinity on-target cellular definition
EC50
Affinity on-target cellular assay type
Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 mins by scintillation counting
Affinity on-target cellular relation
=