Compound name
Telmisartan
Protein family
GPCR
Target name
AGTR2
Affinity biochemical (nM)
0.33
Compound EUbOPEN ID
EUB0000415a
SMILES
CCCC1=NC2=C(C)C=C(C=C2N1CC1=CC=C(C=C1)C1=CC=CC=C1C(O)=O)C1=NC2=CC=CC=C2N1C
InChIKey
RMMXLENWKUUMAY-UHFFFAOYSA-N
NCBI gene ID
186
UniProt ID
P50052
Synonyms
AT2, MRX88
Mode of action
Antagonist
Affinity biochemical definition
IC50
Affinity biochemical assay type
Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma counting
Affinity Biochemical Source Knowledge
22309912
Affinity biochemical relation
=