Compound name
ZM-241385
Protein family
GPCR
Target name
ADORA2A
Affinity biochemical (nM)
0.92
Affinity on-target cellular (nM)
1.39
Compound EUbOPEN ID
EUB0000417a
SMILES
NC1=NC(NCCC2=CC=C(O)C=C2)=NC2=NC(=NN12)C1=CC=CO1
InChIKey
PWTBZOIUWZOPFT-UHFFFAOYSA-N
NCBI gene ID
135
UniProt ID
P29274
Synonyms
RDC8
Mode of action
Antagonist
Affinity biochemical definition
Ki
Affinity biochemical assay type
Binding affinity towards human Adenosine A2a receptor expressed in HEK293 cells using 6 nM [3H]CGS-21680
Affinity Biochemical Source Knowledge
16250647
Affinity biochemical relation
=
Affinity on-target cellular definition
Ki
Affinity on-target cellular assay type
Inhibition of human recombinant adenosine receptor A2a
Affinity on-target cellular relation
=