Compound name
CGP-12177
Protein family
GPCR
Target name
ADRB1
Affinity on-target cellular (nM)
12.3
Compound EUbOPEN ID
EUB0000420aCl
SMILES
[H]Cl.CC(C)(C)NCC(O)COC1=C2NC(=O)NC2=CC=C1
InChIKey
YQVFCYCTITZLSX-UHFFFAOYSA-N
NCBI gene ID
153
UniProt ID
P08588
Affinity on-target cellular definition
EC50
Affinity on-target cellular assay type
Partial agonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrs
Affinity on-target cellular relation
=