Compound name
CGP-12177
Protein family
GPCR
Target name
ADRB2
Affinity biochemical (nM)
1.95
Compound EUbOPEN ID
EUB0000420aCl
SMILES
[H]Cl.CC(C)(C)NCC(O)COC1=C2NC(=O)NC2=CC=C1
InChIKey
YQVFCYCTITZLSX-UHFFFAOYSA-N
NCBI gene ID
154
UniProt ID
P07550
Synonyms
ADRBR, BAR, B2AR
Mode of action
Antagonist
Affinity biochemical definition
Kd
Affinity biochemical assay type
Displacement of [3H]DHA from inactive/G protein-uncoupled human beta2-AR expressed in CHO cell membranes by liquid scintillation counting
Affinity Biochemical Source Knowledge
27239696
Affinity biochemical relation
=