Compound name
PLERIXAFOR
Protein family
GPCR
Target name
CCR2
Affinity biochemical (nM)
0.06
Compound EUbOPEN ID
EUB0000474aCl
SMILES
[H]Cl.C(N1CCCNCCNCCCNCC1)C1=CC=C(CN2CCCNCCNCCCNCC2)C=C1
InChIKey
VZVSLNRDUPMOSZ-UHFFFAOYSA-N
NCBI gene ID
729230
UniProt ID
P41597
Synonyms
CC-CKR-2, CKR2, MCP-1-R, CD192, FLJ78302
Mode of action
Antagonist
Affinity biochemical definition
IC50
Affinity biochemical assay type
Displacement of [125I]MCP1 from CCR2/CXCR4 expressed in CHOK1 cells
Affinity Biochemical Source Knowledge
17715128
Affinity biochemical relation
=