Compound name
INDACATEROL
Protein family
GPCR
Target name
ADRB2
Affinity biochemical (nM)
39.35
Affinity on-target cellular (nM)
10.96
CG-Set
Not included in the set
Compound EUbOPEN ID
EUB0000499a
SMILES
CCC1=CC2=C(CC(C2)NC[C@H](O)C2=C3C=CC(=O)NC3=C(O)C=C2)C=C1CC
InChIKey
QZZUEBNBZAPZLX-QFIPXVFZSA-N
NCBI gene ID
154
UniProt ID
P07550
Synonyms
ADRBR, BAR, B2AR
Mode of action
Agonist
Affinity biochemical definition
Ki
Affinity biochemical assay type
Displacement of [125I]cyanopindolol from human recombinant beta2 adrenergic receptor expressed in CHO cells by filtration assay
Affinity Biochemical Source Knowledge
20402514
Affinity biochemical relation
=
Affinity on-target cellular definition
EC50
Affinity on-target cellular assay type
Agonist activity at human beta2 adrenergic receptor assessed as increase in cAMP level by whole cell assay
Affinity on-target cellular relation
=