Compound name
NIBR0213
Protein family
GPCR
Target name
S1PR1
Affinity on-target cellular (nM)
2
Compound EUbOPEN ID
EUB0000501a
SMILES
C[C@H](NC(=O)C1=C(C)C=C(C=C1C)C1=CC(N[C@H](C)C2=CC(C)=C(Cl)C=C2)=CC=C1)C(O)=O
InChIKey
KYHUARFFBDLROH-MOPGFXCFSA-N
NCBI gene ID
1901
UniProt ID
P21453
Synonyms
edg-1, D1S3362, CD363
Mode of action
Antagonist
Affinity on-target cellular definition
IC50
Affinity on-target cellular assay type
Antagonist activity at human S1P1 receptor expressed in CHO cells after 120 mins by [35S]GTPgammaS binding assay
Affinity on-target cellular relation
=