Compound name
GSK106
Protein family
Hydrolase
Target name
PADI4
Affinity biochemical (nM)
100000
CG-Set
Other targets
Recommended Concentration
1 µM
Compound EUbOPEN ID
EUB0001070aCl
SMILES
CCn1c(-c2nc3cc(C(=O)N4CC[C]C(N)C4)ccc3n2C)cc2ccccc21.[Cl]
InChIKey
PLCVQSIOQUTHPT-UHFFFAOYSA-N
NCBI gene ID
23569
UniProt ID
Q9UM07
Synonyms
PAD, PAD4, PADI5, PDI4, PDI5
Mode of action
Negative control for GSK484
Affinity biochemical definition
IC50
Affinity biochemical assay type
Fluorescence polarization binding assay (0 mM Ca)
Affinity Biochemical Source Knowledge
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4397581/
Affinity biochemical relation
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