Compound name
NI-198
Protein family
Bromodomain
Target name
BRPF3
Affinity biochemical (nM)
100000
CG-Set
Epigenetic set
Recommended Concentration
1 µM
Compound EUbOPEN ID
EUB0001074a
SMILES
O=S(NC1=CC=C2N(C(C(CC)=CC2=C1)=O)CC)(C3=CC=C(C=C3)C#N)=O
InChIKey
QTIVTZLLONAWRR-UHFFFAOYSA-N
NCBI gene ID
27154
UniProt ID
Q9ULD4
Synonyms
KIAA1286
Mode of action
BRPF3@BRD
Affinity biochemical definition
IC50
Affinity biochemical assay type
BROMOscan
Affinity Biochemical Source Knowledge
https://pubs.acs.org/doi/10.1021/acs.jmedchem.7b00611#
Affinity biochemical relation
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