Compound name
NVS-PAK1-C
Protein family
Protein Kinase
Target name
PAK1
Affinity biochemical (nM)
1500
CG-Set
Kinase set
Recommended Concentration
1 µM
Compound EUbOPEN ID
EUB0001075a
SMILES
O=C(N1CC[C@@H](C1)NC2=NC3=C(N(C4=C2C=C(Cl)C=C4)CC(F)F)C=CC(F)=C3)N(C)C
InChIKey
RVHZFZVJXGIAJF-HNNXBMFYSA-N
NCBI gene ID
5058
UniProt ID
Q13153
Mode of action
Negative control for NVS-PAK1-1
Affinity biochemical definition
IC50
Affinity biochemical assay type
Caliper in-vitro dephosphorylation assay (PAK1 phos.)
Affinity Biochemical Source Knowledge
https://www.thesgc.org/chemical-probes/mu1742
Affinity biochemical relation
=