Compound name
MU2027
Protein family
Protein Kinase
Target name
CSNK1D
Affinity biochemical (nM)
3000
Affinity on-target cellular (nM)
50000
CG-Set
Kinase set
Recommended Concentration
1 µM
Compound EUbOPEN ID
EUB0001201a
SMILES
CCc1ccc(-c2ncn(CC3(F)CCN(C)CC3)c2-c2ccnc3[nH]ccc23)nc1
InChIKey
SRSOVGVHVNSXTC-UHFFFAOYSA-N
NCBI gene ID
1453
UniProt ID
P48730
Synonyms
HCKID, CKID, CKIdelta
Mode of action
Negative control for MU1742
Affinity biochemical definition
IC50
Affinity biochemical assay type
Tracer competition assays (Reaction Biology, 10 mM ATP)
Affinity Biochemical Source Knowledge
https://www.thesgc.org/chemical-probes/mu1742
Affinity biochemical relation
>
Affinity on-target cellular definition
IC50
Affinity on-target cellular assay type
NanoBRET asssay (HEK293T cells)
Affinity on-target cellular source knowledge
https://www.thesgc.org/chemical-probes/mu1742
Affinity on-target cellular relation
>