Compound name
SGC-CDKL5/GSK3-1N
Protein family
Protein Kinase
Target name
GSK3B
Affinity on-target cellular (nM)
10000
CG-Set
Kinase set
Recommended Concentration
100 nM
Compound EUbOPEN ID
EUB0002313a
SMILES
Cn1cc(NC(=O)c2cc(F)cc(F)c2)c(C(=O)NC2CCNCC2)n1
InChIKey
ODZBDODDFLVDQZ-UHFFFAOYSA-N
NCBI gene ID
2932
UniProt ID
P49841
Mode of action
Negative control for SGC-CDKL5_GSK3
Affinity on-target cellular definition
IC50
Affinity on-target cellular assay type
NanoBRET assay (HEK293T cells)
Affinity on-target cellular source knowledge
https://www.thesgc.org/chemical-probes/SGC-CDKL5_GSK3
Affinity on-target cellular relation
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